1354819-22-9Relevant articles and documents
The discovery of tetrahydropyridine analogs as hNav1.7 selective inhibitors for analgesia
Wu, Wentao,Li, Zhixiang,Yang, Guangwen,Teng, Mingxing,Qin, Jian,Hu, Zhijing,Hou, Lijuan,Shen, Liang,Dong, Haiheng,Zhang, Yang,Li, Jian,Chen, Shuhui,Tian, Jingwei,Zhang, Jianzhao,Ye, Liang
, p. 2210 - 2215 (2017)
hNav1.7 small molecular inhibitors have attracted lots of attention by its unique analgesic effect. Herein, we report the design and synthesis of a novel series of tetrahydropyridine analogs as hNav1.7 inhibitors for analgesia. Detail structural–activity