135964-76-0Relevant academic research and scientific papers
DERIVATIZED 3-STYRYL-CEPHALOSPORINS
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, (2014/10/18)
Broad spectrum beta-lactamase inhibitors. Certain inhibitors also exhibit potent antibiotic activity in addition to beta-lactamase inhibition. Compounds of the invention are designed such that on cleavage of the beta-lactam ring reactive moieties are generated which can inactivate beta-lactamase. Also provided are methods of making betalactamase inhibitors and beta-lactam antibiotics exhibiting such inhibition. Additionally provided are pharmaceutical compositions for treatment or prevention of bacterial infections and methods of treatment of such infections.
Novel phenylalanine derivatives
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Page/Page column 42, (2010/02/14)
Specific phenylalanine derivatives and analogues thereof have an antagonistic activity to α4 integrin. They are used as therapeutic agents for various diseases concerning α4 integrin.
QUINAZOLINE DERIVATIVES AND THEIR PREPARATION
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, (2008/06/13)
A compound of the formula: STR1 in which R 1 and R 2 are each hydrogen, halogen, nitro, amino, protected amino, hydroxyamino, lower alkyl, hydroxy, protected hydroxy, sulfamoyl, carboxy, protected carboxy, mercapto, optionally substituted heterocyclic-car
Quinazoline derivatives
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, (2008/06/13)
Compounds of the formula: STR1 are described wherein R 1, R 2, R 3 and A are described in the claims. These compounds show significant dopamine receptor agonist activity.
