1360066-72-3Relevant articles and documents
SELECTIVE GRP94 INHIBITORS AND USES THEREOF
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Paragraph 0215; 0220, (2015/02/25)
The disclosure relates to novel selective Grp94 inhibitors, compositions comprising an effective amount of such compounds, and methods to treat or prevent a condition, such as cancer, comprising administering to an animal in need thereof an effective amount of such compounds.
An efficient copper-catalyzed microwave-assisted S-arylation towards the synthesis of 8-arylsulfanyl adenines
Sun, Weilin,Patel, Pallav D.,Stephani, Ralph A.,Chiosis, Gabriela
experimental part, p. 3008 - 3012 (2012/01/05)
We report a microwave-assisted synthetic protocol for the C-S cross-coupling reaction of aryl iodides and 8-mercaptoadenine using CuI and n-Bu4NBr with NaOt-Bu in DMF. The method is rapid, simple, and cost efficient, and leads in high yields to