1361550-95-9Relevant academic research and scientific papers
A diverted total synthesis of mycolactone analogues: An insight into buruli ulcer toxins
Chany, Anne-Caroline,Casarotto, Virginie,Schmitt, Marjorie,Tarnus, Celine,Guenin-Mace, Laure,Demangel, Caroline,Mirguet, Olivier,Eustache, Jacques,Blanchard, Nicolas
, p. 14413 - 14419 (2011)
Mycolactones are complex macrolides responsible for a severe necrotizing skin disease called Buruli ulcer. Deciphering their functional interactions is of fundamental importance for the understanding, and ultimately, the control of this devastating mycobacterial infection. We report herein a diverted total synthesis approach of mycolactones analogues and provide the first insights into their structure-activity relationship based on cytopathic assays on L929 fibroblasts. The lowest concentration inducing a cytopathic effect was determined for selected analogues, allowing a clear picture to emerge by comparison with the natural toxins.
STRUCTURAL VARIANTS OF MYCOLACTONES FOR USE IN MODULATING INFLAMMATION, IMMUNITY AND PAIN
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, (2013/06/05)
The present invention is related to variants of mycolactones of formula (I), processes for the preparation thereof, pharmaceutical compositions thereof and their use in modulating inflammation, immunity and pain. Y-O-W (I), wherein Y and W are as defined in claim 1.
Structural variants of mycolactones for use in modulating inflammation, immunity and pain
-
, (2013/06/05)
The present invention is related to variants of mycolactones of formula (I), processes for the preparation thereof, pharmaceutical compositions thereof and their use in modulating inflammation, immunity and pain. ???????? Y-O-W?????(I) wherein Y and W are as defined in claim 1.
