1363411-87-3Relevant academic research and scientific papers
The p-toluenesulfonic acid-catalyzed transformation of polyfluorinated 2-alkynylanilines to 2-aminoarylketones and indoles
Politanskaya, Larisa,Shteingarts, Vitalij,Tretyakov, Evgeny,Potapov, Alexander
supporting information, p. 5328 - 5332 (2015/09/01)
The reactivity of a series of polyfluorinated 2-alkynylanilines with various alcohols using p-TSA has been studied. It was found that hydration of the triple bond gave rise to polyfluorinated 2-aminoarylketones and competed with an electrophilic heterocyc
Synthesis of polyfluorinated ortho-alkynylanilines
Politanskaya, Larisa V.,Chuikov, Igor P.,Kolodina, Ekaterina A.,Shvartsberg, Mark S.,Shteingarts, Vitalij D.
, p. 97 - 107 (2012/03/27)
A series of polyfluorinated ortho-alkynylanilines - the versatile building blocks for diverse polyfluorobenzo azaheterocycles - have been synthesized by the Sonogashira reaction of polyfluorinated ortho-iodanilines with terminal alkynes.
