1366180-75-7Relevant academic research and scientific papers
Discovery of 4-hydroxy-1,6-naphthyridine-3-carbonitrile derivatives as novel PDE10A inhibitors
Bauer, Udo,Giordanetto, Fabrizio,Bauer, Martin,O'Mahony, Gavin,Johansson, Kjell E.,Knecht, Wolfgang,Hartleib-Geschwindner, Judith,Carlsson, Eva T?ppner,Enroth, Cristofer
supporting information; experimental part, p. 1944 - 1948 (2012/04/17)
A series of 1,6-naphthyridine-based compounds was synthesized as potent phosphodiesterase 10A (PDE10A) inhibitors. Structure-based chemical modifications of the discovered chemotype served to further improve potency and selectivity over DHODH, laying the foundation for future optimization efforts.
