138716-17-3Relevant academic research and scientific papers
A one-pot sequential five-component domino reaction for the expedient synthesis of polysubstituted pyrroles
Ambethkar, Sethurajan,Padmini, Vediappen,Bhuvanesh, Nattamai
, p. 4705 - 4709 (2016)
A series of novel pyrrole derivatives has been synthesized from readily available acetophenone, N,N-dimethylformamide dimethyl acetal, aniline, arylglyoxal and malononitrile in methanol under reflux conditions. This one-pot reaction constitutes a new and
Synthesis, in vitro, and in vivo (Zebra fish) antitubercular activity of 7,8-dihydroquinolin-5(6H)-ylidenehydrazinecarbothioamides
Kantevari, Srinivas,Krishna, Vagolu Siva,Marvadi, Sandeep kumar,Sridhar, Balasubramanian,Srilakshmi Reshma, Rudraraju,Sriram, Dharmarajan,Surineni, Goverdhan
, (2020/02/04)
We, herein, describe the synthesis of a series of novel aryl tethered 7,8-dihydroquinolin-5(6H)-ylidenehydrazinecarbothioamides 4a–v, which showed in vitro and in vivo antimycobacterial activity against Mycobacterium tuberculosis (Mtb) H37Rv. The intermed
Pd-catalyzed site selective C-H acetoxylation of aryl/heteroaryl/thiophenyl tethered dihydroquinolinones
Patpi, Santhosh Reddy,Sridhar, Balasubramanian,Tadikamalla, Prabhakar Rao,Kantevari, Srinivas
, p. 10251 - 10261 (2013/09/02)
Described herein is an efficient protocol for the site selective oxidative C-H activation/acetoxylation of a series of 2-aryl/heteroaryl/thiophenyl tethered dihydroquinolinones using palladium acetate as the catalyst and iodobenzene diacetate as an oxidan
Synthesis and antimicrobial activity of novel 7-(Heteroaryl)-1,2,4- triazolo[1,5-a]-pyrimidine derivatives
Rama Rao, R. Janaki,Rao, A.K.S. Bhujanga,Swapna,Rani, B. Baby,Murthy
experimental part, p. 1837 - 1843 (2012/08/07)
The synthesis, characterization and antimicrobial activity of novel 1,2,4-triazolo[1,5-a]pyrimidines have been reported. The compounds were prepared by acid catalyzed condensation of 3-amino-1,2,4-triazole with 3-(dialkylamino)acryloalkanone.
Synthesis and antitubercular evaluation of novel substituted aryl and thiophenyl tethered dihydro-6H-quinolin-5-ones
Kantevari, Srinivas,Patpi, Santhosh Reddy,Sridhar, Balasubramanian,Yogeeswari, Perumal,Sriram, Dharmarajan
scheme or table, p. 1214 - 1217 (2011/04/16)
A series of novel aryl and thiophenyl tethered dihydro-6H-quinolin-5-ones have been synthesized in very good yields through CeCl3· 7H2O-NaI catalyzed one-pot condensation of β-enaminones derived from the respective methyl ketones; 1,
Synthesis and antibacterial activity of novel 5-(heteroaryl)isoxazole derivatives
RamaRao, R. Janaki,Rao, A.K.S. Bhujanga,Sreenivas,Kumar, B. Suneel,Murthy
experimental part, p. 243 - 250 (2011/06/26)
The synthesis, characterization and antibacterial activity of novel isoxazole derivatives were reported. 3-Di (alkylamino)acryloalkanones were prepared and used as synthons to get the target isoxazole derivatives via reaction with hydroxylamine hydrochloride or hydroxylamine-O-sulphonic acid.
Facile diversity-oriented synthesis and antitubercular evaluation of novel aryl and heteroaryl tethered pyridines and dihydro-6H-quinolin-5-ones derived via variants of the Bohlmann-Rahtz reaction
Kantevari, Srinivas,Patpi, Santhosh Reddy,Addla, Dinesh,Putapatri, Siddamal Reddy,Sridhar, Balasubramanian,Yogeeswari, Perumal,Sriram, Dharmarajan
experimental part, p. 427 - 435 (2011/09/14)
The diversity oriented synthesis of substituted pyridines and dihydro-6H-quinolin-5-ones tethered with aryls and heteroaryls was achieved in very good yields through CeCl3?7H2O-NaI catalyst via variants of the Bohlmann-Rahtz reaction
SUBSTITUTED THIOPHENE DERIVATIVES AS ANTI-CANCER AGENTS
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Page/Page column 116-117, (2008/06/13)
The present invention relates to new substituted five-membered compounds and pharmaceutically acceptable salts, esters or prodrugs thereof, compositions of the new compounds together with pharmaceutically acceptable carriers, and uses of the new compounds
