1391088-46-2Relevant articles and documents
Thiorhodamines containing amide and thioamide functionality as inhibitors of the ATP-binding cassette drug transporter P-glycoprotein (ABCB1)
Orchard, Alexandra,Schamerhorn, Gregory A.,Calitree, Brandon D.,Sawada, Geri A.,Loo, Tip W.,Claire Bartlett,Clarke, David M.,Detty, Michael R.
, p. 4290 - 4302 (2012)
Twelve thiorhodamine derivatives have been examined for their ability to stimulate the ATPase activity of purified human P-glycoprotein (P-gp)-His 10, to promote uptake of calcein AM and vinblastine into multidrug-resistant, P-gp-overexpressing