1395047-49-0Relevant articles and documents
Identification and characterization of diarylimidazoles as hybrid inhibitors of butyrylcholinesterase and amyloid beta fibril formation
Karlsson, Daniela,Fallarero, Adyary,Brunhofer, Gerda,Guzik, Przemyslaw,Prinz, Michaela,Holzgrabe, Ulrike,Erker, Thomas,Vuorela, Pia
experimental part, p. 169 - 183 (2012/04/23)
In this contribution, a chemical collection of aromatic compounds was screened for inhibition on butyrylcholinesterase (BChE)'s hydrolase activity using Ellman's reaction. A set of diarylimidazoles was identified as highly selective inhibitors of BChE hyd