1398089-68-3Relevant academic research and scientific papers
Discovery of liver selective non-steroidal glucocorticoid receptor antagonist as novel antidiabetic agents
Shah, Kiran,Patel, Dipam,Jadav, Pradip,Sheikh, Mubeen,Sairam, Kalapatapu V. V. M.,Joharapurkar, Amit,Jain, Mukul R.,Bahekar, Rajesh
, p. 5857 - 5862,6 (2020/07/31)
Series of benzyl-phenoxybenzyl amino-phenyl acid derivatives (8a-q) are reported as non-steroidal GR antagonist. Compound 8g showed excellent h-GR binding and potent antagonistic activity (in vitro). The lead compound 8g exhibited significant oral antidia
