1402242-65-2Relevant academic research and scientific papers
Synthesis of ynone trifluoroborates toward functionalized pyrazoles
Kirkham, James D.,Edeson, Steven J.,Harrity, Joseph P. A.,Stokes, Stephen
, p. 5354 - 5357,4 (2012/12/12)
The synthesis of a range of novel ynone trifluoroborates has been achieved, in a two-pot process from propargylic alcohols. These alkynes have been subsequently used in the formation of a range of pyrazole trifluoroborate salts via cyclization with hydrazines. The products are generated with high levels of regiocontrol and in excellent yields and represent versatile synthetic intermediates.
