1404307-40-9Relevant academic research and scientific papers
An efficient synthesis of 3-substituted N-glycoside indoles useful as sodium-dependent glucose transporter inhibitors
Li, Xun,Wells, Kenneth M.,Branum, Shawn,Damon, Sandra,Youells, Scott,Beauchamp, Derek A.,Palmer, David,Stefanick, Stephen,Russell, Ronald K.,Murray, William
, p. 1727 - 1732 (2013/01/15)
A practical synthesis of two N-glycoside indoles 1 and 2, identified as highly potent sodium-dependent glucose transporter (SGLT) inhibitors is described. Highlights of the synthetic process include a selective and quantitative Vilsmeier acylation and a h
