141543-20-6Relevant articles and documents
Synthesis of 2-phosphonoheterocycles via base-promoted 5-endo cyclization
Bousbia, Ameni,Benkhoud, Mohamed Lamine,El-Ka?m, Laurent,Prévost, Sébastien
supporting information, (2021/01/14)
Herein, a synthesis of 2-phosphonodihydrofurans and 2-phosphonodihydropyrroles via 5-endo cyclization of O-and N-propargylated compounds is described. The reaction is promoted by potassium tert-butoxide and allows a fast access to interesting heterocycles which were easily converted into 2-arylated pyrroles under acidic conditions.