1421315-92-5Relevant academic research and scientific papers
Enantioselective synthesis of azaflavanones using organocatalytic 6-endo aza-Michael addition
Cheng, Shuanghua,Zhao, Lili,Yu, Shouyun
, p. 982 - 986 (2014/04/03)
A method to prepare highly enantioenriched azaflavanones using an organocatalytic 6-endo aza-Michael addition has been described. A variety of 2-aryl-, 2-vinyl- and 2-methylazaflavanones were prepared in good yields (53-84%) and excellent enantioselectivities (97.6:2.4 to 99.3:0.7 er).
Asymmetric Bronsted acid-catalyzed intramolecular aza-michael reaction - Enantioselective synthesis of dihydroquinolinones
Rueping, Magnus,Moreth, Stefan A.,Bolte, Michael
, p. 1021 - 1029 (2013/01/15)
The enantioselective synthesis of 2-aryl-substituted 2,3-dihydroquinolin-4- ones, a class of heterocyclic compounds with interesting biological activities, has been achieved through a Bronsted acidcatalyzed enantioselective intramolecular Michael addition. The products are available in moderate to high yields and with good enantioselectivities.
