1421689-79-3Relevant academic research and scientific papers
Short and efficient route toward α-substituted N-arylazetidines from acetanilides via Mitsunobu reaction
Kern, Nicolas,Hoffmann, Marie,Weibel, Jean-Marc,Pale, Patrick,Blanc, Aurélien
, p. 5519 - 5531 (2015/03/30)
N-Arylazetidines are efficiently obtained in a three-step procedure, providing a wide diversity of derivatives on multigram scale with overall yields of 21-55%. Cheap or easily available acetanilides are used in an adapted aldolization with aldehydes, fur
Gold(I)-catalyzed rearrangement of N-aryl 2-alkynylazetidines to pyrrolo[1,2-a]indoles
Kern, Nicolas,Hoffmann, Marie,Blanc, Aurelien,Weibel, Jean-Marc,Pale, Patrick
, p. 836 - 839 (2013/03/29)
Various N-aryl-2-alkynylazetidines were very efficiently converted to pyrrolo[1,2-a]indoles with gold catalysts, especially the 2-biphenyl- dicyclohexylphosphino-gold(I) hexafluoroantimonate, in dichloromethane at room temperature. Additionally, two forma
