1421781-90-9Relevant academic research and scientific papers
A concise synthesis of N-substituted fagomine derivatives and the systematic exploration of their α-glycosidase inhibition
Jiang, Fu-Xiang,Liu, Qiao-Zhen,Zhao, Dan,Luo, Cui-Ting,Guo, Cui-Ping,Ye, Wen-Cai,Luo, Cheng,Chen, Heru
, p. 211 - 222 (2014/04/03)
A novel and concise scheme has been developed successfully for the syntheses of N-substituted fagomine derivatives. The transformation of lactone (2) to 1,5-diol (3) was carried on with high yield (93-95%). The cyclization of 4 to 5 is a high stereoselect
