1427310-62-0Relevant articles and documents
Amino acid derived quinazolines as Rock/PKA inhibitors
Chowdhury, Sarwat,Chen, Yen Ting,Fang, Xingang,Grant, Wayne,Pocas, Jennifer,Cameron, Michael D.,Ruiz, Claudia,Lin, Li,Park, Hajeung,Schr?ter, Thomas,Bannister, Thomas D.,Lograsso, Philip V.,Feng, Yangbo
, p. 1592 - 1599 (2013/04/10)
SAR and lead optimization studies for Rock inhibitors based on amino acid-derived quinazolines are described. Studies demonstrated that these amino acid derived quinazolinones were mainly pan-Rock (I & II) inhibitors. While selectivity against other kinas