142958-94-9Relevant academic research and scientific papers
One-Pot N-Arylation of indoles directly from N-arylsulfonylindoles via consecutive deprotection and SnAr reactions with activated aryl halides
Xu, Hui,Fan, Ling-Ling
experimental part, p. 321 - 323 (2009/11/30)
An efficient one-pot step by step t-BuOK-mediated procedure for the synthesis of N-arylindoles has been developed in moderate to good yields. The protocol involves the consecutive deprotection of N-arylsulfonylindoles as latent indoles and subsequent SnAr
Indole- and benzimidazole-substituted imidazole and benzimidazole derivatives
-
, (2008/06/13)
Novel compounds are disclosed having the formula STR1 wherein X, R1, R2, R3, R4, and R5 are substituents. These compounds inhibit the action of angiotensin II and are useful, therefore, for example, as antihypertensive agents.
