1443511-06-5Relevant academic research and scientific papers
Synthesis and anticancer activity of dichloroplatinum(II) complexes of podophyllotoxin
Liu, Xuan,Zhang, Lin-Lin,Xu, Xiao-Hui,Hui, Lin,Zhang, Jin-Bang,Chen, Shi-Wu
supporting information, p. 3780 - 3784 (2013/07/27)
A series of dichloroplatinum(II) complexes of podophyllotoxin (PPT) were prepared, and their cytotoxicity against sensitive (A-549, HeLa, HCT-8, Hep-G2, K562) and resistant (ADM/K562) cell lines were evaluated. Complex cis-[4α-O-(2″,3″-diaminopropanoyl)-podophyllotoxin] dichloride platinum(II) (12) displayed most potent cytotoxicity with IC50 value in the range 0.071-2.98 μM. Complex 12 induces cell cycle arrest in the G2/M phase, and inhibits the formation of microtubules in HeLa cells. Furthermore, this complex exhibits potent DNA cleavage capabilities.
