1450759-38-2Relevant academic research and scientific papers
Synthesis of potent CERT inhibitor HPA-12 featuring a tandem corey-link and intramolecular nucleophilic acyl substitution reaction
Snider, Jason R.,Entrekin, Jordan T.,Snowden, Timothy S.,Dolliver, Debra
supporting information, p. 1899 - 1903 (2013/07/26)
A novel preparation of the potent CERT protein inhibitor (1R,3S)-HPA-12 is described. The synthesis is accomplished in five steps from (S)-Wynberg lactone and features a diastereoselective tandem Corey-Link and intramolecular nucleophilic acyl substitution reaction in a key step. Georg Thieme Verlag Stuttgart · New York.
