145878-51-9Relevant articles and documents
BENZODIAZEPINE DERIVATIVES, COMPOSITIONS CONTAINING THEM AND THEIR USE IN THERAPY
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, (2008/06/13)
Compounds of Formula (I), and salts and prodrugs thereof wherein: R. sup.1 is H, certain optionally substituted C 1-6 alkyl or C 3-7 cycloalkyl; R 2 represents a group (a) wherein X is O, S or NR 8 where R 8 is H or C 1-4 alkyl; one of Z and Y is C= O and the other is O, S or NR 9, where R 9 is H or C 1-4 alkyl; R 3 is C 1-6 alkyl, halo or NR 6 R 7 ; R 4 is C 3-10 cycloalkyl; n is 0, 1, 2 or 3, and are CCK and/or gastrin antagonists, which compounds and compositions thereof are useful in therapy.