146714-63-8Relevant articles and documents
Synthesis and evaluation of 4-(2'-methoxyphenyl)-1-[2'-[N-(2''- pyridinyl)-p-iodobenzamido]ethyl]piperazine (p-MPPI): A new iodinated 5- HT(1A) ligand [2]
Zhuang,Kung,Kung
, p. 1406 - 1407 (1994)
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Structural Insights into 5-HT1A/D4 Selectivity of WAY-100635 Analogues: Molecular Modeling, Synthesis, and in Vitro Binding
Dilly, Sébastien,Liégeois, Jean-Fran?ois
, p. 1324 - 1331 (2016/08/02)
The resurgence of interest in 5-HT1A receptors as a therapeutic target requires the existence of highly selective 5-HT1A ligands. To date, WAY-100635 has been the prototypical antagonist of these receptors. However, this compound als
NOVEL SYNTHESIS METHOD
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Page/Page column 17, (2013/04/10)
The present invention relates to a method of making compounds having affinity for the 1 A subtype of the serotonin receptor, i.e. 5HT1A. The method of the present invention provides advantages over the known methods of synthesis. The compounds