146953-22-2Relevant academic research and scientific papers
Synthesis of conformationally constrained macrocyclic analogs of the potent and selective CCK-B antagonist CI-988
Bolton,Roth,Trivedi
, p. 525 - 536 (2007/10/02)
A series of conformationally constrained analogs of the potent CCK-B antagonist CI-988 were prepared and evaluated for their CCK-B binding affinity. A macrolactamization reaction leading to the conformation of 11 to 14-membered rings was also investigated
