147440-64-0Relevant academic research and scientific papers
Synthesis of novel triazol compounds containing isatin as potential antibacterial and antifungal agents by microwave and conventional methods
Oezil, Musa,Mentese, Emre,Yilmaz, Fatih,Islamoglu, Fatih,Kahveci, Bahittin
, p. 268 - 271 (2011)
Microwave irradiation has been used to accelerate the conversion of isatin (1a) and 5-nitroisatin (1b) into their Schiff bases 3-[5′-aryl(alkyl)- 2′,4′-dihydro-1′,2′,4′-triazol-3′-on- 4′-yl]iminoisatin (3a-g) and 3-[5′-aryl(alkyl)-2′,4′- dihydro-1′,2′,4′-triazol-3′-on-4′-yl] imino-5-nitroisatin (4a-g), respectively. Reaction was achieved by microwave-induced technique, which reduced the reaction time drastically and improved the yield when compared to conventional heating. The newly synthesised bases showed moderate antimicrobial activity against the standard bacterial and fungal organisms tested.
Synthesis, in vitro antimicrobial and antioxidant activities of some new 4,5-dihydro-1h-1,2,4-triazol-5-one derivatives
Yueksek, Haydar,Akyildirim, Onur,Yola, Mehmet L.,Guersoy-Kol, Oezlem,Celebier, Mustafa,Kart, Didem
, p. 470 - 480 (2013)
A series of compounds derived from 4,5-dihydro-1H-1,2,4-triazol-5-one were synthesized and characterized by spectral data. The 12 new compounds were analyzed for their potential in vitro antioxidant activities by three different methods. Compound 4f showe
Synthesis and in vitro antioxidant and antimicrobial activities of novel 3-alkyl(aryl)-4-[3-methoxy-4-(2-furylcarbonyloxy)-benzylidenamino]-4,5-dihydro-1H-1,2,4-triazol-5-ones, and their N-acetyl, N-Mannich base derivatives
Manap, Sevda
, (2021/09/03)
The reactions of 3-alkyl(aryl)-4-amino-4,5-dihydro-1H-1,2,4-triazol-5-ones (1) with 3-methoxy-4-(2-furylcarbonyloxy)-benzaldehyde (2) formed 3-alkyl(aryl)-4-[3-methoxy-4-(2-furylcarbonyloxy)-benzylidenamino]-4,5-dihydro-1H-1,2,4-triazol-5-ones (3). Moreov
In vitro antioxidant and antimicrobial properties of some new 4,5-dihydro-1H-1,2,4-triazole-5-ones
Akta?-Yoku?,Yüksek,Gürsoy-Kol,Alpay-Karao?lu
, p. 389 - 396 (2018/09/29)
In this study, 3-alkyl(aryl)-4-amino-4,5-dihydro-1H-1,2,4-triazol-5-ones (3a-3h) reacted with 3-benzenesulfonyloxy-4-methoxybenzaldehyde (1a-1h) to afford eight new 3-alkyl(aryl)-4-(3-benzenesulfonyloxy-4-methoxybenzylidenamino)-4,5-dihydro-1H-1,2,4-triaz
Study of antioxidant properties and DNA interaction of some novel 4,5-Dihydro-1H-1,2,4-triazol-5-one derivatives
Arslantas, Ali,Yüksek, Haydar,Gürsoy-Kol, ?zlem,Ocak, Zafer,Tomruk, Zeynep,Calapoglu, Mustafa
scheme or table, p. 3327 - 3334 (2012/07/28)
3-Alkyl(aryl)-4-amino-4,5-dihydro-1H-1,2,4-triazol-5-ones (2) reacted with 4-benzenesulfonyloxybenzaldehyde (3) to afford the corresponding seven novel 3-alkyl(aryl)-4-(4-benzenesulfonyloxybenzylidenamino)-4,5-dihydro-1H-1,2, 4-triazol-5-ones (4). The ace
Synthesis and in-vitro antioxidant evaluation of some novel 4-(4-substituted) benzylidenamino-4,5-dihydro-1H-1,2,4-triazol-5-ones
Yueksek, Haydar,Guersoy-Kol, Oezlem,Kemer, Guel,Ocak, Zafer,Anil, Baris
, p. 325 - 330 (2013/09/24)
3-Alkyl (aryl)-4-amino-4,5-dihydro-1H-1,2,4-triazol-5-ones (2a-g) were reacted with 4-ethylbenzaldehyde to afford the corresponding 3-alkyl (aryl).4-(4-ethylbenzylidenamino)-4,5-dihydro-1H-1,2.4-triazol-5-ones (3a-g). The acetylation reactions of compound
Synthesis and in vitro antioxidant evaluation of some novel 4, 5-dihydro-1h-1, 2, 4-triazol-5-one derivatives
Gursoy Kol,Yuksek
experimental part, p. 123 - 136 (2011/01/03)
In this study, thirteen novel 4,5-dihydro-1H-1,2,4-triazol-5-one derivatives were synthesized and characterized by elemental analyses and IR, 1H NMR,13C NMR and UV spectral data. The synthesized compounds were analyzed for their in v
Determination of the protonation constants of some 4-(substituted benzylamino)-4,5-dihydro-1H-1,2,4-triazol-5-ones by the potentiometric method in ethanol-water mixtures
Islamoglu, Fatih,Kahveci, Bahittin,Islamoglu, Yahya
, p. 36 - 41 (2008/09/17)
To gain more information about the effect of solvent on 4,5-dihydro-1H-1,2,4-triazol-5-ones, the stoichiometric protonation constants of thirteen triazoles in ethanol-water mixtures were determined at an ionic strength of 0.10MNaCl and at 25.0 ± 0.1°C und
Synthesis and antitumor activities of some 4,5-dihydro-1H-1,2,4-triazol-5-ones
Ikizler, Aykut A.,Ikizler, Aysun,Serdar, Mevluet,Yildirim, Nuri
, p. 363 - 370 (2007/10/03)
Eight new 3-alkyl(aryl)-4-arylidenamino-4,5-dihydro-1H-1,2,4-triazol-5-ones were synthesized and characterised by elemental analysis, 1H NMR, IR and UV spectra. Seven new and 34 recently reported derivatives of 4,5-dihydro-1H-1,2,4-triazol-5-one ring were screened for their antitumor activities.
