14819-39-7Relevant articles and documents
Chemo- and regioselective synthesis of alkyl-3-thiazoline carboxylates
Fernandez, Xavier,Fellous, Roland,Lizzani-Cuvelier, Louisette,Loiseau, Michel,Duach, Elisabet
, p. 1519 - 1521 (2001)
The synthesis of a series of allyl substituted 3-thiazoline-carboxylates was carried out from the corresponding thiazolidines, by a MnO2-mediated oxidation reaction under mild conditions. The reaction was chemoselective towards the amine-imine oxidation and was also regioselective, affording the unsaturation at the 3-position of the heterocycle.
Oxidation of 4-carboxylate thiazolines to 4-carboxylate thiazoles by molecular oxygen
Huang, Yue,Gan, Haifeng,Li, Shang,Xu, Jinyi,Wu, Xiaoming,Yao, Hequan
supporting information; experimental part, p. 1751 - 1753 (2010/05/18)
A facile and environment-benign oxidation by molecular oxygen was applied for the conversion of 4-carboxylate thiazolines to 4-carboxylate thiazoles. The substituent effect on thiazoline ring was investigated. It was found that electron-poor group on the thiazoline ring could facilitate the oxidation.
TETRACYCLIC COMPOUNDS AS DOPAMINE AGONISTS
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, (2008/06/13)
A tetracyclic compound of the formula: STR1 wherein A and the atoms to which it is attached and the optional double bond represent a mono-or di-heterocyclic ring selected from: STR2 wherein R 1, R. sup.2, R 3, R 4 and X are specifically defined, which compounds are useful in the treatment of dopamine-related neurological, psychological and cardiovascular disorders as well as in the treatment of substance abuse and other addictive behavior disorders, cognitive impairment and attention deficit disorder.