150689-77-3Relevant academic research and scientific papers
Benzodiazepine derivatives, compositions containing them and their use in therapy
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, (2008/06/13)
Compounds of formula (I), and salts and prodrugs thereof STR1 wherein: R 1 is H, certain optionally substituted C 1-6 alkyl, or C 3-7 cyclocalkyl;R 2 represents a group STR2 wherein X is O, S or NR 8 where R 8 is H or C 1-4 alkyl; R 3 is C 1-6 alkyl, halo or NR 6 R 7 ;R 4 is C 1-7 alkyl, C 3-7 cycloalkyl, C 4-7 cycloalkylalkyl or optionally substituted aryl;n is 0, 1, 2 or 3; are CCK and/or gastrin receptor antagonists. They and compositions thereof are useful in therapy.
