153484-02-7Relevant articles and documents
Potent Gastrin-Releasing Peptide (GRP) Antagonists Derived from GRP (19-27) with a C-Terminal DProΨPhe-NH2 and N-Terminal Aromatic Residues
Leban, Johann J.,Landavazo, Antonio,McDermed, John D.,Diliberto, Emanuel J.,Jansen, Marilyn,et al.
, p. 439 - 445 (1994)
We have previously reported that octapeptides with a -DProΨPhe-NH2 C-terminus are potent GRP antagonists and have greatly enhanced in vivo stability.Now we report the detailed syntheses of such peptides and additional attempts to further increase m