153560-02-2Relevant academic research and scientific papers
Regioselective three-component synthesis of 1,2-diarylindoles from cyclohexanones, α-hydroxyketones and anilines under transition-metal-free conditions
Li, Cheng,Xie, Yanjun,Xiao, Fuhong,Huang, Huawen,Deng, Guo-Jun
supporting information, p. 4079 - 4082 (2019/04/25)
A facile method for the one-pot synthesis of 1,2-diarylindoles under transition-metal-free conditions is described. Cyclohexanones were used as the aryl sources via the dehydrogenative aromatization process. One C-C and two C-N bonds were selectively formed via a domino reaction. This protocol provides a convenient approach for the construction of valuable bioactive 1,2-diarylindoles from readily available cyclohexanones, α-hydroxyketones and anilines.
Iodine-mediated α-sulfonyloxylation of alkyl aryl ketones with oxone and sulfonic acids
Kikui, Hiroki,Moriyama, Katsuhiko,Togo, Hideo
, p. 791 - 797 (2013/04/10)
Alkyl aryl ketones are converted into the corresponding α-sulfonyloxyketones, in moderate to excellent yields, via a novel procedure that utilizes Oxone, p-toluenesulfonic acid or methanesulfonic acid and molecular iodine in a mixture of aceton
Bridgehead Nitrogen Heterocycles: Facile Synthesis of Imidazo -1,3,4-Thiadiazoles Using Hypervalent Iodine
Mohan, Jag,Singh, Virender,Kataria, Sangeeta
, p. 617 - 619 (2007/10/03)
2,6 Diarylimidazo -1,3,4 thiadiazoles (3) were synthesized by reactions of either α-haloketones with 2-aminothiadiazoles (1) or directly with acetophenones in the presence of benzene.The latter method is convenient and vers
