155204-28-7Relevant articles and documents
Structural Insights into 5-HT1A/D4 Selectivity of WAY-100635 Analogues: Molecular Modeling, Synthesis, and in Vitro Binding
Dilly, Sébastien,Liégeois, Jean-Fran?ois
, p. 1324 - 1331 (2016/08/02)
The resurgence of interest in 5-HT1A receptors as a therapeutic target requires the existence of highly selective 5-HT1A ligands. To date, WAY-100635 has been the prototypical antagonist of these receptors. However, this compound als
NOVEL SYNTHESIS METHOD
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Page/Page column 32-33, (2013/04/10)
The present invention relates to a method of making compounds having affinity for the 1 A subtype of the serotonin receptor, i.e. 5HT1A. The method of the present invention provides advantages over the known methods of synthesis. The compounds
EFFICIENT SYNTHETIC METHOD OF 18F-MEFWAY PRECURSOR
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Page/Page column 8, (2012/06/16)
The present invention relates a novel method for preparing an 18F-mefway precursor. The present invention provides an efficient synthetic method of an 18F-mefway precursor, which comprises an improved the acid chloride coupling react