155381-86-5Relevant academic research and scientific papers
Macrocyclic Renin Inhibitors: Synthesis of A Subnanomolar, Orally Active Cysteine Derived Inhibitor
Yang, Lihu,Weber, Ann E.,Greenlee, William J.,Patchett, Arthur A.
, p. 7035 - 7038 (2007/10/02)
A class of novel thioether linked macrocyclic renin inhibitors was synthesized.A key element of the synthesis is the use of boroxazolidone for the simultaneous protection of the amino and carboxyl groups in L-cysteine.
