1558029-00-7Relevant academic research and scientific papers
In vitro membrane permeation studies and in vivo antinociception of glycosylated Dmt1-DALDA analogues
Ballet, Steven,Betti, Cecilia,Novoa, Alexandre,Toemboely, Csaba,Uhd Nielsen, Carsten,Helms, Hans Christian,Lesniak, Anna,Kleczkowska, Patrycja,Chung, Nga N.,Lipkowski, Andrzej W.,Brodin, Birger,Tourwe, Dirk,Schiller, Peter W.
, p. 352 - 357 (2014/05/06)
In this study the μ opioid receptor (MOR) ligands DALDA (Tyr-d-Arg-Phe-Lys-NH2) and Dmt1-DALDA (Dmt-d-Arg-Phe-Lys-NH2, Dmt = 2′,6′-dimethyltyrosine) were glycosylated at the N- or C-terminus. Subsequently, the modified pep
