156997-88-5Relevant academic research and scientific papers
Synthesis of Nb-acyltryptamines and their 1-hydroxy-tryptamine derivatives as new α2-blockers
Yamada, Koji,Tanaka, Yoshio,Somei, Masanori
experimental part, p. 635 - 645 (2009/12/26)
Nb-Acyl- and Nb-acyl-1-hydroxytryptamines are found to be novel and structurally simple (α2-blocker for the treatment of erectile dysfunction.
Synthesis and structure - Activity relationships of novel naphthalenic and bioisosteric related amidic derivatives as melatonin receptor ligands
Leclerc, Veronique,Fourmaintraux, Eric,Depreux, Patrick,Lesieur, Daniel,Morgan, Peter,Howell, H. Edward,Renard, Pierre,Caignard, Daniel-Henri,Pfeiffer, Bruno,Delagrange, Philippe,Guardiola-Lemaitre, Beatrice,Andrieux, Jean
, p. 1875 - 1887 (2007/10/03)
A previous paper reported the synthesis of melatonin receptor ligands. In order to complete the structure-activity relationships and to obtain antagonists to the melatonin receptor, a new series of naphthalenic analogues of melatonin have been synthesized
