1594796-75-4Relevant academic research and scientific papers
The direct C-H halogenations of indoles
Shi, Leilei,Zhang, Dongmei,Lin, Riyuan,Zhang, Chun,Li, Xun,Jiao, Ning
supporting information, p. 2243 - 2245 (2014/04/17)
A novel and efficient transition metal-free C-H bond halogenation of indole derivatives has been developed. 3-Halogenated (3-Br, 3-I) indoles are highly regioselectively produced by this protocol. Simple and readily available halide salts (TBAB, KI) are employed as the halogen source. The transition metal-free and the mild conditions make this protocol very easy to handle and practical.
