1607788-95-3Relevant articles and documents
Preliminary investigations into triazole derived androgen receptor antagonists
Altimari, Jarrad M.,Niranjan, Birunthi,Risbridger, Gail P.,Schweiker, Stephanie S.,Lohning, Anna E.,Henderson, Luke C.
, p. 2692 - 2706 (2014/05/06)
A range of 1,4-substituted-1,2,3-N-phenyltriazoles were synthesized and evaluated as non-steroidal androgen receptor (AR) antagonists. The motivation for this study was to replace the N-phenyl amide portion of small molecule antiandrogens with a 1,2,3-tri