1608474-90-3Relevant articles and documents
Discovery of azaisoerianin derivatives as potential antitumors agents
Soussi, Mohamed Ali,Provot, Olivier,Bernadat, Guillaume,Bignon, Jérome,Wdzieczak-Bakala, Joanna,Desravines, Déborah,Dubois, Jo?lle,Brion, Jean-Daniel,Messaoudi, Samir,Alami, Mouad
, p. 178 - 189 (2014/04/17)
A series of N-methyl-diarylamines 2 was designed and synthesized as a novel class of CA-4 and isoCA-4 analogues. Compounds 2b and 2m showed excellent antiproliferative activity with mean GI50 values at a nanomolar level in a diverse set of huma