1609205-22-2Relevant academic research and scientific papers
Tandem synthesis of 4-aminoxanthones is controlled by a water-assisted tautomerization: a general straightforward reaction
Bornadiego, Ana,Díaz, Jesús,Marcos, Carlos F.
supporting information, p. 1410 - 1422 (2019/02/14)
Aminoxanthones constitute a group of therapeutically promising compounds that so far have been synthetically challenging. Here, we report the synthesis of both aminodihydroxanthones and fully aromatized aminoxanthones by an easy to perform, one-step multi
Synthesis of 4-aminoxanthones by an uncatalyzed, multicomponent reaction
Bornadiego, Ana,Diaz, Jesus,Marcos, Carlos F.
, p. 718 - 722 (2014/04/03)
The synthesis of xanthones via a multicomponent reaction of isocyanides is described for the first time. In this one-pot process, a tandem [4+1] plus [4+2] cycloaddition leads to polysubstituted 4-aminoxanthones in excellent to quantitative yields at room temperature in a non-catalyzed reaction.
