1610892-93-7Relevant academic research and scientific papers
New series of sulfonamides containing amino acid moiety act as effective and selective inhibitors of tumor-associated carbonic anhydrase XII
Ceruso, Mariangela,Bragagni, Marco,Alothman, Zeid,Osman, Sameh M.,Supuran, Claudiu T.
, p. 430 - 434 (2015/07/27)
New benzenesulfonamides incorporating water solubilizing moieties were synthesized using N-α-acetyl-l-lysine or γ-aminobutyric acid as scaffolds followed by the conversion of their terminal amino group to the guanidine one. Their inhibition activity was a
Sulfonamides with potent inhibitory action and selectivity against the α-carbonic anhydrase from Vibrio cholerae
Ceruso, Mariangela,Del Prete, Sonia,Alothman, Zeid,Capasso, Clemente,Supuran, Claudiu T.
supporting information, p. 826 - 830 (2014/08/05)
By using N-α-acetyl-l-lysine or GABA scaffolds and the conversion of the terminal amino group to the guanidine one, benzenesulfonamides incorporating water solubilizing moieties were synthesized. The new compounds were medium potency inhibitors of the cyt
