1619929-45-1Relevant articles and documents
Pyrrole–aminopyrimidine ensembles: Cycloaddition of guanidine to acylethynylpyrroles
Budaev, Arsalan B.,Ivanov, Andrey V.,Petrova, Olga V.,Sagitova, Elena F.,Sobenina, Lyubov N.,Trofimov, Boris A.,Ushakov, Igor A.
, (2021/06/16)
An efficient method for the synthesis of pharmaceutically prospective pyrrole–aminopyrimidine ensembles (in up to 91% yield) by the cyclocondensation of easily available acylethynylpyrroles with guanidine nitrate has been developed. The reaction proceeds
From 4,5,6,7-tetrahydroindoles to 3- or 5-(4,5,6,7-tetrahydroindol-2-yl) isoxazoles in two steps: A regioselective switch between 3- and 5-isomers
Sobenina, Lyubov N.,Tomilin, Denis N.,Gotsko, Maxim D.,Ushakov, Igor A.,Mikhaleva, Albina I.,Trofimov, Boris A.
, p. 5168 - 5174 (2014/07/08)
(4,5,6,7-Tetrahydroindol-2-yl)alkynes, synthesized by cross-coupling of 4,5,6,7-tetrahydroindoles with aroyl(hetaroyl)bromoalkynes or ethyl bromopropynoate in the presence of K2CO3, regioselectively cyclize with hydroxylamine to eith