1620006-80-5Relevant articles and documents
Highly enantioselective aza-Henry reaction with isatin N-Boc ketimines
Holmquist, Melireth,Blay, Gonzalo,Pedro, José R.
, p. 9309 - 9312 (2014)
A highly enantioselective aza-Henry reaction with isatin N-Boc ketimines using a Cu(ii)-BOX complex as a catalyst is described. The reaction, which does not require protection of the N1 atom, provides the corresponding nitroamines bearing a quaternary stereocentre with high yields and enantiomeric excesses (up to 99.9%).