1632196-79-2Relevant academic research and scientific papers
Copper-catalyzed N-arylation of azoles and diazoles using highly functionalized trivalent organobismuth reagents
Petiot, Pauline,Dansereau, Julien,Gagnon, Alexandre
, p. 22255 - 22259 (2014/06/23)
The N-arylation of indoles, indazoles, pyrroles, and pyrazoles using highly functionalized trivalent arylbismuth reagents is reported. The reaction is promoted by a substoichiometric amount of copper acetate, and it tolerates a wide diversity of functional groups on the azole and the organobismuth reagent. The method is also applied to the N-arylation of tryptophan derivatives. This journal is the Partner Organisations 2014.
