167770-27-6Relevant articles and documents
4,10-Dihydro-5H-thieno[3,2-c][1]benzazepine derivatives and 9,10- dihydro-4H-thieno[2,3-c][1]benzazepine derivatives as orally active arginine vasopressin receptor antagonists
Aranapakam, Venkatesan,Albright, J. Donald,Grosu, George T.,Chan, Peter S.,Coupet, Joseph,Saunders, Trina,Ru, Xun,Mazandarani
, p. 1733 - 1736 (2007/10/03)
Synthesis and structure-activity relationships (SAR) of arginine vasopressin receptor (AVP) antagonists are described. Potent and orally active compounds are prepared when tricyclic 10,11-dihydro-5H-pyrrolo[2,1- c][1,4]benzodiazepine moiety in VPA-985 1 i
Tricyclic benzazepine oxytocin and vasopressin antagonists.
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, (2008/06/13)
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Preparation of tricyclic benzazepine vasopressin antagonists.
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, (2008/06/13)
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