168030-60-2Relevant academic research and scientific papers
Three-component synthesis of N-boc-4-iodopyrroles and sequential one-pot alkynylation
Merkul, Eugen,Boersch, Christina,Frank, Walter,Mueller, Thomas J.J.
supporting information; experimental part, p. 2269 - 2272 (2009/09/30)
(Hetero)aryl-, alkenyl-, and selected alkyl-substituted acid chlorides can be efficiently coupled with N-Boc-protected propargylamine to produce ynones which are converted in a one-pot fashion to 2-substituted N-Boc-4-iodopyrroles. Upon addition of a furt
