17337-81-4

Upstream product

• 17327-71-8 N^α-Benzyloxycarbonyl-N^γ-tert.-Butoxycarbonyl-L-2,4-diamino-butyryl-Phe-amid 
• 849948-77-2 (1'S, 2S)-4-(N-Boc-amino)-N'-(1'-carbamoyl-2'-phenylethyl)-2-(N''-Fmoc-amino)butanamide 
• 5241-58-7 L-Phenylalanine amide 

Downstream Products

• 849948-78-3 4-(N-Boc-amino)-N'-((S)-1-carbamoyl-2-phenylethyl)-(S)-2-(N''-(4-methyl-1-naphthalenesulfonyl)amino)butanamide 

Relevant academic research and scientific papers

SOMATOSTATIN RECEPTOR 1 AND/OR 4 SELECTIVE AGONISTS AND ANTAGONISTS

The invention relates to (hetero)arylsulfonylamino based peptidomimetics of formula (I), wherein R1, R2, R3, A, B, D, Q, k and n are defined as disclosed, or a pharmaceutically acceptable salt or ester thereof. Compounds of formula (I) possess high affinity and selectivity for the somatostatin receptor subtypes SSTR1 and/or SSTR4 and can be used for the treatment or diagnosis of diseases or conditions wherein an interaction with SSTR1 and/or SSTR4 is indicated to be useful.