174174-72-2Relevant academic research and scientific papers
Synthesis and in vitro activities of highly potent and selective tripeptide antagonists of the neurokinin NK-1 receptor
Caliendo,Greco,Grieco,Perissutti,Santagada,Calignano,Mancuso,Novellino
, p. 755 - 759 (2007/10/03)
We report on the synthesis and the pharmacological properties of a new series of tachykinin antagonists based on the tripeptide Ac-Thr-D-Trp(CHO)-Phe-N(Me)-Bzl (1, FR113680) partly modified on the C-terminal amide part. Stereochemistry around the benzilic
