1743-90-4Relevant academic research and scientific papers
ARYL SULFAMIDE DERIVATIVES AND METHODS OF THEIR USE
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Page/Page column 124, (2008/12/06)
The present invention is directed to aryl sulfamide derivatives of formula (I): or a pharmaceutically acceptable salt, stereoisomer or tautomer thereof, which are monoamine reuptake inhibitors, compositions containing these derivatives, and methods of their use for the prevention and treatment of conditions, including, inter alia, vasomotor symptoms, sexual dysfunction, gastrointestinal disorders and genitourinary disorder, depression disorders, endogenous behavioral disorders, cognitive disorders, diabetic neuropathy, pain, and other diseases or disorders.
Novel 1,5-benzodiazepines as CCK-B ligands. Effect of aryl-carbamic substituents at the C-3 position together with halogen substitution on the benzo-fused ring
Tranquillini, M. Elvira,Cassara, Paolo G.,Corsi, Mauro,Curotto, Giovanni,Donati, Daniele,Finizia, Gabriella,Pentassuglia, Giorgio,Polinelli, Stefano,Tarzia, Giorgio,Ursini, Antonella,Van Amsterdam, Franciscus T.M.
, p. 353 - 357 (2007/10/03)
The synthesis and biological evaluation as potential CCK-B receptor ligands of a number of 1-isopentyl-3-aryloxycarbamoyl-5-aryl-1,5-benzodiazepines substituted with halogen atoms on the benzo-fused ring is here briefly discussed.
