176965-99-4Relevant articles and documents
Synthesis of A-79175: A second generation 5-lipoxygenase inhibitor
Dickman, Daniel A.,Ku, Yi-Yin,Morton, Howard E.,Chemburkar, Sanjay R.,Patel, Hemantkumar H.,Thomas, Albert,Plata, Daniel J.,Sawick, David P.
, p. 1791 - 1795 (2007/10/03)
A convergent, high yielding, and scalable synthesis of A-79175, with a key step involving a mild and efficient Cu-Pd catalyzed coupling reaction of a terminal acetylene with a substituted 2-iodofuran is discussed.
