178034-81-6Relevant articles and documents
Synthesis and structure-activity relationships of 2-substituted D-tryptophan-containing peptidic endothelin receptor antagonists: Importance of the C-2 substituent of the D-tryptophan residue for endothelin A and B receptor subtype selectivity
Fukami, Takehiro,Yamakawa, Takeru,Niiyama, Kenji,Kojima, Hisaki,Amano, Yuuka,Kanda, Fuyuko,Ozaki, Satoshi,Fukuroda, Takahiro,Ihara, Masaki,Yano, Mitsuo,Ishikawa, Kiyofumi
, p. 2313 - 2330 (2007/10/03)
Continuing studies on modifications of potent cyclic pentapeptide endothelin (ET) receptor antagonists, represented by BQ-123, and potent linear tripeptide derivative ET receptor antagonists, represented by BQ-788, are described herein. The introduction o