192717-41-2Relevant articles and documents
Potent nonpeptide GnRH receptor antagonists derived from substituted indole-5-carboxamides and -acetamides bearing a pyridine side-chain terminus
Ashton, Wallace T.,Sisco, Rosemary M.,Yang, Yi Tien,Lo, Jane-Ling,Yudkovitz, Joel B.,Gibbons, Patrice H.,Mount, George R.,Ren, Rena Ning,Butler, Bridget S.,Cheng, Kang,Goulet, Mark T.
, p. 1727 - 1731 (2007/10/03)
A pyridine side-chain terminus has been incorporated into the indole-5-carboxamide and indole-5-acetamide series of GnRH antagonists. Potent activity was observed in binding and functional assays. Certain branched or cyclic tertiary amides were identified