197568-73-3Relevant academic research and scientific papers
A Short Stereocontrolled Synthesis of Hydroxyethylene Dipeptide Isosteres
Jones, D. Michael,Nilsson, Bo,Szelke, Michael
, p. 2286 - 2290 (2007/10/02)
A stereocontrolled synthesis of protected hydroxyethylene dipeptide isosteres 14 and 16 is described.It provides the 2R,4S,5S epimers required for the preparation of aspartic proteinase inhibitors.The choice of a benzene ring as a precursor to the carboxy
