198553-25-2Relevant articles and documents
Novel piperidinylpyrimidine derivatives as inhibitors of HIV-1 LTR activation
Fujiwara, Norio,Nakajima, Takashi,Ueda, Yutaka,Fujita, Hitoshi,Kawakami, Hajime
experimental part, p. 9804 - 9816 (2009/04/06)
Piperidinylpyrimidine derivatives, previously prepared as inhibitors of TNF-α production, were evaluated for their inhibitory activity against HIV-1 LTR activation. Some of these derivatives inhibited activation of HIV-1 LTR-directed CAT gene expression i